IACS-9571 - CAS# 1800477-30-8 size:10mg solid 7 nM and 14 nM

7 nM and 14 nM

FIDAS-5 has anticancer activities

Chemical Name: 1-Methyl-7-nitro-2H-3

59865-13-3

G9a functions as a molecular scaffold for assembly of transcriptional coactivators on a subset of glucocorticoid receptor target genes

IACS-9571 - CAS# 1800477-30-8 size:10mg solid 7 nM and 14 nMIACS 9571, CAS No. 1800477 30 8, is a potent and selective inhibitor TRIM24 and BRPF1. IACS 9571 has low nanomolar affinities for TRIM24 and BRPF1 (ITC Kd = 31 nM and 14 nM, respectively). With its excellent cellular potency (EC50 = 50 nM) and favorable pharmacokinetic properties (F = 29%), IACS 9571 is a high quality chemical probe for the evaluation of TRIM24 and or BRPF1 bromodomain function in vitro and in vivo. Product information CAS Number: